Hispidulin

CAS No. 1447-88-7

Hispidulin( —— )

Catalog No. M21669 CAS No. 1447-88-7

Hispidulin a natural flavone with a broad spectrum of biological activities is a Pim-1 inhibitor (IC50: 2.71 μM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 49 Get Quote
2MG 29 Get Quote
5MG 46 Get Quote
10MG 73 Get Quote
25MG 120 Get Quote
50MG 174 Get Quote
100MG 254 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Hispidulin
  • Note
    Research use only, not for human use.
  • Brief Description
    Hispidulin a natural flavone with a broad spectrum of biological activities is a Pim-1 inhibitor (IC50: 2.71 μM).
  • Description
    Hispidulin a natural flavone with a broad spectrum of biological activities is a Pim-1 inhibitor (IC50: 2.71 μM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    JAK/STAT Signaling
  • Target
    Pim
  • Recptor
    Pim1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1447-88-7
  • Formula Weight
    300.27
  • Molecular Formula
    C16H12O6
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 60 mg/mL (199.82 mM; Need ultrasonic);Water: Insoluble
  • SMILES
    COc(c(O)c(c(OC(c(cc1)ccc1O)=C1)c2)C1=O)c2O
  • Chemical Name
    57-Dihydroxy-2-(4-hydroxyphenyl)-6-methoxychromen-4-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Chao SW et al. Total Synthesis of Hispidulin and the Structural Basis for Its Inhibition of Proto-oncogene KinasePim-1. J Nat Prod. 2015 Aug 28;78(8):1969-76.
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