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Dermorphin
CAS No. 77614-16-5
Dermorphin( —— )
Catalog No. M20802 CAS No. 77614-16-5
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 46 | In Stock |
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| 5MG | 93 | In Stock |
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| 10MG | 158 | In Stock |
|
| 25MG | 316 | In Stock |
|
| 50MG | 536 | In Stock |
|
| 100MG | 791 | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameDermorphin
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NoteResearch use only, not for human use.
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Brief DescriptionDermorphin is agonist of μ-opioid receptor (MOR) agonist.
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DescriptionDermorphin is agonist of μ-opioid receptor (MOR) agonist.
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In VitroDermorphin, a peptide isolated from the skin of Phyllomedusa frogs and the peptide receptor (NOP) component by the endogenous agonist nociceptin/orphanin FQ (N/OFQ). In displacement binding studies at CHOhMu, Dermorphin and DeNo displac the binding of [3H]-DPN in a concentration dependent and saturable manner. Dermorphin displays an affinity of 7.17, while N/OFQ fails to displace [3H]-DPN at the Delta receptor. Dermorphin and DeNo stimulate the binding of GTPγ[35S] in a concentration dependent and saturable manner at the Mu receptor.
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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Recptorμ-opioid receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number77614-16-5
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Formula Weight802.87
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Molecular FormulaC40H50N8O10
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Purity>98% (HPLC)
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SolubilityIn Vitro:?H2O : 120 mg/mL (149.46 mM)
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SMILESCC(NC(=O)C(N)Cc1ccc(O)cc1)C(=O)NC(Cc1ccccc1)C(=O)NCC(=O)NC(Cc1ccc(O)cc1)C(=O)N1CCCC1C(=O)NC(CO)C(N)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Robinson M A Guan F Mcdonnell S et al. Pharmacokinetics and pharmacodynamics of dermorphin in the horse[J]. Journal of Veterinary Pharmacology and Therapeutics 2015 38(4):321-329.
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