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NMDAR antagonist 1
CAS No. 2220162-06-9
NMDAR antagonist 1( —— )
Catalog No. M20173 CAS No. 2220162-06-9
NMDAR antagonist 1 is a potent and orally bioavailable NR2B-selective antagonist of NMDAR.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 98 | In Stock |
|
| 10MG | 155 | In Stock |
|
| 25MG | 297 | In Stock |
|
| 50MG | 416 | In Stock |
|
| 100MG | 551 | In Stock |
|
| 200MG | 728 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameNMDAR antagonist 1
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NoteResearch use only, not for human use.
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Brief DescriptionNMDAR antagonist 1 is a potent and orally bioavailable NR2B-selective antagonist of NMDAR.
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DescriptionNMDAR antagonist 1 is a potent and orally bioavailable NR2B-selective antagonist of NMDAR.
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In VitroNMDAR antagonist 1 (Compound 5q) exhibits excellent neuroprotective activity. NMDAR antagonist 1 can attenuate Ca2+ influx induced by NMDA.NMDAR antagonist 1 can suppress the NR2B up-regulation and increase p-ERK1/2 expression.NMDAR antagonist 1 inhibits SH-SY5Y cells with cell viabilities of 75.8%, 80.0%, 84.4%, and 78.6% at 0.1 μM 1 μM 10 μM 100 μM, respectively.
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorOthers
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Research Area——
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Indication——
Chemical Information
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CAS Number2220162-06-9
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Formula Weight414.3
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Molecular FormulaC20H20BrN3O2
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Purity>98% (HPLC)
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Solubility——
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SMILESCc1ccc2N=C3CCC(N3Cc2c1)C(=O)NCCc1ccc(O)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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