Cart
sales@molnova.com
NMDAR antagonist 1
CAS No. 2220162-06-9
NMDAR antagonist 1( —— )
Catalog No. M20173 CAS No. 2220162-06-9
NMDAR antagonist 1 is a potent and orally bioavailable NR2B-selective antagonist of NMDAR.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 98 | In Stock |
|
| 10MG | 155 | In Stock |
|
| 25MG | 297 | In Stock |
|
| 50MG | 416 | In Stock |
|
| 100MG | 551 | In Stock |
|
| 200MG | 728 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameNMDAR antagonist 1
-
NoteResearch use only, not for human use.
-
Brief DescriptionNMDAR antagonist 1 is a potent and orally bioavailable NR2B-selective antagonist of NMDAR.
-
DescriptionNMDAR antagonist 1 is a potent and orally bioavailable NR2B-selective antagonist of NMDAR.
-
In VitroNMDAR antagonist 1 (Compound 5q) exhibits excellent neuroprotective activity. NMDAR antagonist 1 can attenuate Ca2+ influx induced by NMDA.NMDAR antagonist 1 can suppress the NR2B up-regulation and increase p-ERK1/2 expression.NMDAR antagonist 1 inhibits SH-SY5Y cells with cell viabilities of 75.8%, 80.0%, 84.4%, and 78.6% at 0.1 μM 1 μM 10 μM 100 μM, respectively.
-
In Vivo——
-
Synonyms——
-
PathwayOthers
-
TargetOther Targets
-
RecptorOthers
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2220162-06-9
-
Formula Weight414.3
-
Molecular FormulaC20H20BrN3O2
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCc1ccc2N=C3CCC(N3Cc2c1)C(=O)NCCc1ccc(O)cc1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
molnova catalog
related products
-
(Pro3)-Dynorphin A (...
(Pro3)-Dynorphin A (1-11) amide
-
Deapi-platycodin D3
Deapi-platycodin D3 is a natural product isolate from the root of Platycodon grandiflorum.
-
(R)-5-Hydroxy-1,7-di...
(R)-5-Hydroxy-1,7-diphenylheptan-3-one is extracted from the rhizomes of Alpinia officinarum, a Chinese medicinal herb. (R)-5-Hydroxy-1,7-diphenylheptan-3-one inhibits melanogenesis in theophylline-stimulated murine B16 melanoma 4A5 cells.
