Bepridil hydrochloride

CAS No. 68099-86-5

Bepridil hydrochloride( CERM 1978 )

Catalog No. M20140 CAS No. 68099-86-5

Bepridil is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX) sodium channels and cardiac sarcolemmal KATP channels.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 28 In Stock
10MG 38 In Stock
25MG 77 In Stock
50MG 105 In Stock
100MG 152 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Bepridil hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Bepridil is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX) sodium channels and cardiac sarcolemmal KATP channels.
  • Description
    Bepridil is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX) sodium channels and cardiac sarcolemmal KATP channels.(In Vitro):Bepridil hydrochloride is a calcium channel blocker, with antianginal activity.(In Vivo):Bepridil hydrochloride (21 mg/kg) reduces heart rate and mean arterial pressure, decreases the mean coronary vascular resistance and increases stroke volume in rats.
  • In Vitro
    Bepridil hydrochloride is a calcium channel blocker, with antianginal activity.
  • In Vivo
    Bepridil hydrochloride (21 mg/kg) reduces heart rate and mean arterial pressure, decreases the mean coronary vascular resistance and increases stroke volume in rats.
  • Synonyms
    CERM 1978
  • Pathway
    GPCR/G Protein
  • Target
    Calcium Channel
  • Recptor
    Calcium Channel
  • Research Area
    Cardiovascular Disease
  • Indication
    Angina pectoris; Tachycardia

Chemical Information

  • CAS Number
    68099-86-5
  • Formula Weight
    403
  • Molecular Formula
    C24H35ClN2O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 130 mg/mL (322.58 mM)
  • SMILES
    Cl.CC(C)COCC(CN(Cc1ccccc1)c1ccccc1)N1CCCC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Flaim SF et al. Effects of bepridil hydrochloride on cardiocirculatory dynamics coronary vascular resistance and cardiac output distribution in normal conscious rats. J Cardiovasc Pharmacol. 1988 Mar;11(3):363-72.
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