mTOR inhibitor-1

CAS No. 468747-17-3

mTOR inhibitor-1( —— )

Catalog No. M20101 CAS No. 468747-17-3

C-4 is a potential ATP-competitive inhibitor of mTOR. C-4 could inhibit cell growth and proliferation.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 31 In Stock
5MG 50 In Stock
10MG 84 In Stock
25MG 170 In Stock
50MG 267 In Stock
100MG 444 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    mTOR inhibitor-1
  • Note
    Research use only, not for human use.
  • Brief Description
    C-4 is a potential ATP-competitive inhibitor of mTOR. C-4 could inhibit cell growth and proliferation.
  • Description
    C-4 is a potential ATP-competitive inhibitor of mTOR. C-4 could inhibit cell growth and proliferation.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    PI3K/Akt/mTOR signaling
  • Target
    mTOR
  • Recptor
    mTOR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    468747-17-3
  • Formula Weight
    363.21
  • Molecular Formula
    C16H15BrN2O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 70 mg/mL (192.72 mM)
  • SMILES
    C\C(=N/NC(=O)c1ccc(C)c(Br)c1)c1ccc(O)cc1O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Liu J et al. In Silico Discovery of a Small Molecule Suppressing Lung Carcinoma A549 Cells Proliferation and Inducing Autophagy via mTOR Pathway Inhibition. Mol Pharm. 2018 Nov 5;15(11):5427-5436.
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