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Imidafenacin

CAS No. 170105-16-5

Imidafenacin( ONO-8025 | KRP-197 )

Catalog No. M19789 CAS No. 170105-16-5

Imidafenacin(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 28 In Stock
25MG 44 In Stock
50MG 66 In Stock
100MG 99 In Stock
200MG 146 In Stock
500MG 250 In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    Imidafenacin
  • Note
    Research use only, not for human use.
  • Brief Description
    Imidafenacin(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.
  • Description
    Imidafenacin(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ONO-8025 | KRP-197
  • Pathway
    Endocrinology/Hormones
  • Target
    AChR
  • Recptor
    mAChR
  • Research Area
    Neurological Disease
  • Indication
    Chronic obstructive pulmonary disease

Chemical Information

  • CAS Number
    170105-16-5
  • Formula Weight
    319.4
  • Molecular Formula
    C20H21N3O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:7.8 mg/mL (24.42 mM) Need ultrasonic and warming
  • SMILES
    Cc1nccn1CCC(C(N)=O)(c1ccccc1)c1ccccc1
  • Chemical Name
    4-(2-Methyl-1-imidazolyl)-22-diphenylbutanamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Yamazaki T et al. Imidafenacin has no influence on learning in nucleus basalis of Meynert-lesioned rats. Naunyn Schmiedebergs Arch Pharmacol. 2013 Dec;386(12):1095-102.
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