Cathepsin Inhibitor 1

CAS No. 225120-65-0

Cathepsin Inhibitor 1( Cathepsin Inhibitor 1 | Cathepsin-Inhibitor-1 | CTS-IN-1 )

Catalog No. M18263 CAS No. 225120-65-0

Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 87 Get Quote
10MG 140 Get Quote
25MG 267 Get Quote
50MG 507 Get Quote
100MG 731 Get Quote
500MG 1503 Get Quote
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Biological Information

  • Product Name
    Cathepsin Inhibitor 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.
  • Description
    Cathepsin Inhibitor 1 is a pan-inhibitor of Cathepsin (L, L2, S, K, B).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Cathepsin Inhibitor 1 | Cathepsin-Inhibitor-1 | CTS-IN-1
  • Pathway
    Immunology/Inflammation
  • Target
    Antiviral
  • Recptor
    Cathepsin K| Cathepsin L| Cathepsin L2| Cathepsin S| Cathepsin S
  • Research Area
    Others-Field
  • Indication
    ——

Chemical Information

  • CAS Number
    225120-65-0
  • Formula Weight
    401.89
  • Molecular Formula
    C20H24ClN5O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (248.82 mM)
  • SMILES
    CN1N=C(C=C1C(=O)N[C@@H](CC1=CC=CC(Cl)=C1)C(=O)NCC#N)C(C)(C)C
  • Chemical Name
    (S)-3-(tert-butyl)-N-(3-(3-chlorophenyl)-1-((cyanomethyl)amino)-1-oxopropan-2-yl)-1-methyl-1H-pyrazole-5-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Asaad N, et al. Bioorg Med Chem Lett, 2009, 19(15), 4280-4283.
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