Protein kinase inhibitors 1

CAS No. 1365986-44-2

Protein kinase inhibitors 1( —— )

Catalog No. M17975 CAS No. 1365986-44-2

Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Protein kinase inhibitors 1
  • Note
    Research use only, not for human use.
  • Brief Description
    Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.
  • Description
    Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Apoptosis
  • Target
    Apoptosis
  • Recptor
    HIPK2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1365986-44-2
  • Formula Weight
    383.42
  • Molecular Formula
    C18H17N5O3S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C4NC(=O)S/C4=C\C=3C=C(c1ccc(nc1)N2CCNCC2)C(=O)NC=3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Miduturu CV, et al. High-throughput kinase profiling: a more efficient approach toward the discovery of new kinaseinhibitors. Chem Biol. 2011 Jul 29;18(7):868-79.
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