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Epinastine HCl
CAS No. 108929-04-0
Epinastine HCl( Epinastine Hydrochloride | Alesion | Elestat )
Catalog No. M17804 CAS No. 108929-04-0
Epinastine is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 37 | In Stock |
|
| 10MG | 31 | In Stock |
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| 25MG | 48 | In Stock |
|
| 50MG | 60 | In Stock |
|
| 100MG | 90 | In Stock |
|
| 200MG | 170 | In Stock |
|
| 500MG | 315 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEpinastine HCl
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NoteResearch use only, not for human use.
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Brief DescriptionEpinastine is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
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DescriptionEpinastine Hydrochloride is a histamine H1 receptor antagonist without sedative activity. Epinastine hydrochloride blocks the histamine H1 receptor and inhibits the release of histamine from mast cells. This prevents the typical allergic symptoms that are caused by histamine activity on capillaries, skin, and mucous membranes. Typical histamine activities include vasodilation, bronchoconstriction, increased vascular permeability, pain, itching, and spasmodic contractions of gastrointestinal smooth muscles. Epinastine HCl also has affinity for histamine H2, 5-HT2, and the alpha-1, alpha-2 adrenergic receptors.
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In Vitro——
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In Vivo——
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SynonymsEpinastine Hydrochloride | Alesion | Elestat
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PathwayOthers
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TargetOther Targets
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RecptorHT
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number108929-04-0
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Formula Weight285.77
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Molecular FormulaC16H15N3·HCl
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Purity>98% (HPLC)
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SolubilityIn Vitro:?H2O : 100 mg/mL (349.93 mM)
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SMILESCl[H].NC1=NCC2N1C1=CC=CC=C1CC1=CC=CC=C21
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Chemical Name3-Amino-9,13b-dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepine Hydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Fügner A, et al. Arzneimittelforschung, 1988, 38(10), 1446-1453.
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