Probimane

CAS No. 108093-90-9

Probimane( Probimane | probimane | AT-2153 | Pro )

Catalog No. M17801 CAS No. 108093-90-9

Probimane had Anti-proliferative effects, cell cycle G2/M phase arrest and blocking of chromosome segregation in human tumor cell lines with MST-16.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 92 In Stock
2MG 33 In Stock
5MG 49 In Stock
10MG 83 In Stock
25MG 198 In Stock
50MG 335 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Probimane
  • Note
    Research use only, not for human use.
  • Brief Description
    Probimane had Anti-proliferative effects, cell cycle G2/M phase arrest and blocking of chromosome segregation in human tumor cell lines with MST-16.
  • Description
    Probimane is anticancer agents. Pro is active against more categories of tumors both in vivo and in vitro, which in some circumstances may make it superior to the currently-used anticancer bisdioxopiperazines, including razoxane and MST-16.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Probimane | probimane | AT-2153 | Pro
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Others
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    108093-90-9
  • Formula Weight
    466.54
  • Molecular Formula
    C21H34N6O6
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(CN1CC(=O)N(C(=O)C1)CN1CCOCC1)N1CC(=O)N(C(=O)C1)CN1CCOCC1
  • Chemical Name
    1-(Morpholin-4-ylmethyl)-4-[2-[4-(morpholin-4-ylmethyl)-3,5-dioxopiperazin-1-yl]propyl]piperazine-2,6-dione

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Lu DY, et al. Anti-proliferative effects, cell cycle G2/M phase arrest and blocking of chromosome segregation by probimane and MST-16 in human tumor cell lines. BMC Pharmacol. 2005 Jun 20;5:11.
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