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MSX-130
CAS No. 4051-59-6
MSX-130( MSX-130 | MSX 130 | MSX130 )
Catalog No. M17502 CAS No. 4051-59-6
MSX-130 is CXCR4 Antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 87 | In Stock |
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| 10MG | 140 | In Stock |
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| 25MG | 267 | In Stock |
|
| 50MG | 500 | In Stock |
|
| 100MG | 705 | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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| 2MG | 33 | In Stock |
|
| 5MG | 51 | In Stock |
|
| 10MG | 87 | In Stock |
|
| 25MG | 188 | In Stock |
|
| 50MG | 305 | In Stock |
|
| 100MG | 477 | In Stock |
|
| 200MG | 677 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMSX-130
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NoteResearch use only, not for human use.
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Brief DescriptionMSX-130 is CXCR4 Antagonist.
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DescriptionMSX-130 is CXCR4 Antagonist.
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In VitroThe C-X-C chemokine receptor-4 (CXCR4) is a seven trans-membrane G-protein coupled receptor (GPCR) classified as a member of the family I GPCR or rhodopsin-like GPCR family. CXCR4 plays an important role in cancer metastasis, regulation of stem cell trafficking, and neovascularization.
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In Vivo——
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SynonymsMSX-130 | MSX 130 | MSX130
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PathwayAutophagy
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TargetCXCR
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RecptorCXCR4
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Research Area——
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Indication——
Chemical Information
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CAS Number4051-59-6
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Formula Weight514
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Molecular FormulaC36H26N4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 2 mg/mL (3.89 mM)
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SMILESc1(ccc(cc1)c1nc(c([nH]1)c1ccccc1)c1ccccc1)c1[nH]c(c(n1)c1ccccc1)c1ccccc1
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Chemical Name2,2'-(1,4-Phenylene)bis[4,5-diphenyl-1H-imidazole]
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Weiqiang Zhan, et al. Discovery of Small Molecule CXCR4 Antagonists. J. Med. Chem., 2007, 50 (23), pp 5655–5664.
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