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Repertaxin

CAS No. 266359-83-5

Repertaxin( Repertaxin | DF 1681Y )

Catalog No. M17461 CAS No. 266359-83-5

Reparixin is a potent inhibitor of both CXCL8 receptors CXCR1/2, it inhibits weakly CXCR2-mediated cell migration (IC50=100 nM), whereas it strongly blocks CXCR1-mediated chemotaxis (IC50=1 nM).

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	107	In Stock
5MG	38	In Stock
10MG	53	In Stock
25MG	117	In Stock
50MG	183	In Stock
100MG	295	In Stock
200MG	439	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

Repertaxin
Note

Research use only, not for human use.
Brief Description

Reparixin is a potent inhibitor of both CXCL8 receptors CXCR1/2, it inhibits weakly CXCR2-mediated cell migration (IC50=100 nM), whereas it strongly blocks CXCR1-mediated chemotaxis (IC50=1 nM).
Description

Reparixin is a potent inhibitor of both CXCL8 receptors CXCR1/2, it inhibits weakly CXCR2-mediated cell migration (IC50=100 nM), whereas it strongly blocks CXCR1-mediated chemotaxis (IC50=1 nM).
In Vitro

——
In Vivo

——
Synonyms

Repertaxin | DF 1681Y
Pathway

GPCR/G Protein
Target

Cannabinoid Receptor
Recptor

CXCR1| CXCR2
Research Area

Inflammation/Immunology
Indication

——

Chemical Information

CAS Number

266359-83-5
Formula Weight

283.39
Molecular Formula

C14H21NO3S
Purity

>98% (HPLC)
Solubility

DMSO : ≥ 500 mg/mL; 1764.35 mM
SMILES

CS(=O)(=O)NC(=O)[C@@H](c1ccc(CC(C)C)cc1)C
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Moriconi A, et al. Design of noncompetitive interleukin-8 inhibitors acting on CXCR1 and CXCR2. J Med Chem. 2007 Aug 23;50(17):3984-4002.

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