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Repertaxin

CAS No. 266359-83-5

Repertaxin( Repertaxin | DF 1681Y )

Catalog No. M17461 CAS No. 266359-83-5

Reparixin is a potent inhibitor of both CXCL8 receptors CXCR1/2, it inhibits weakly CXCR2-mediated cell migration (IC50=100 nM), whereas it strongly blocks CXCR1-mediated chemotaxis (IC50=1 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Repertaxin
  • Note
    Research use only, not for human use.
  • Brief Description
    Reparixin is a potent inhibitor of both CXCL8 receptors CXCR1/2, it inhibits weakly CXCR2-mediated cell migration (IC50=100 nM), whereas it strongly blocks CXCR1-mediated chemotaxis (IC50=1 nM).
  • Description
    Reparixin is a potent inhibitor of both CXCL8 receptors CXCR1/2, it inhibits weakly CXCR2-mediated cell migration (IC50=100 nM), whereas it strongly blocks CXCR1-mediated chemotaxis (IC50=1 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Repertaxin | DF 1681Y
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    CXCR1| CXCR2
  • Research Area
    Inflammation/Immunology
  • Indication
    ——

Chemical Information

  • CAS Number
    266359-83-5
  • Formula Weight
    283.39
  • Molecular Formula
    C14H21NO3S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : ≥ 500 mg/mL; 1764.35 mM
  • SMILES
    CS(=O)(=O)NC(=O)[C@@H](c1ccc(CC(C)C)cc1)C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Moriconi A, et al. Design of noncompetitive interleukin-8 inhibitors acting on CXCR1 and CXCR2. J Med Chem. 2007 Aug 23;50(17):3984-4002.
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