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(R)-Nepicastat HCl

CAS No. 195881-94-8

(R)-Nepicastat HCl( —— )

Catalog No. M17411 CAS No. 195881-94-8

(R)-Nepicastat HCl, the R-enantiomer of Nepicastat HCl, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

(R)-Nepicastat HCl
Note

Research use only, not for human use.
Brief Description

(R)-Nepicastat HCl, the R-enantiomer of Nepicastat HCl, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors.
Description

(R)-Nepicastat HCl, the R-enantiomer of Nepicastat HCl, is a potent and selective inhibitor with IC50 of 25.1 nM and 18.3 nM for bovine and human dopamine-β-hydroxylase, with negligible affinity for twelve other enzymes and thirteen neurotransmitter receptors.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

Dopamine β-hydroxylase| Dopamine β-hydroxylase
Research Area

Cardiovascular Disease
Indication

——

Chemical Information

CAS Number

195881-94-8
Formula Weight

331.81
Molecular Formula

C14H15F2N3S·HCl
Purity

>98% (HPLC)
Solubility

——
SMILES

Cl.NCC1=CNC(=S)N1[C@@H]1CCC2=C(F)C=C(F)C=C2C1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Stanley WC, et al. Br J Pharmacol. 1997, 121(8), 1803-1809.

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