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hnps-PLA Inhibitor
CAS No. 185298-58-2
hnps-PLA Inhibitor( hnps-PLA Inhibitor | MDK-8582 | MDK 8582 )
Catalog No. M17396 CAS No. 185298-58-2
Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 132 | In Stock |
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| 2MG | 70 | In Stock |
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| 5MG | 116 | In Stock |
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| 10MG | 202 | In Stock |
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| 25MG | 341 | In Stock |
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| 50MG | 498 | In Stock |
|
| 100MG | 710 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product Namehnps-PLA Inhibitor
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NoteResearch use only, not for human use.
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Brief DescriptionHnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).
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DescriptionMDK-8582, also known as Hnps-PLA Inhibitor, is an nhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA). The best one inhibited hnps-PLA(2) and LTA(4)H-h with IC(50) values of 9.2 ± 0.5 μM and 2.4 ± 1.4 μM, respectively.
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In Vitro——
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In Vivo——
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Synonymshnps-PLA Inhibitor | MDK-8582 | MDK 8582
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PathwayAngiogenesis
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TargetFGFR
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RecptorLTA(4)H-h| hnsPLA2
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Research Area——
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Indication——
Chemical Information
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CAS Number185298-58-2
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Formula Weight379.42
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Molecular FormulaC21H21N3O4
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(N)C(=O)c1c(CC)n(Cc2ccccc2)c2c1c(OCC(=O)N)ccc2
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Chemical Name2-(4-(2-Amino-2-oxoethoxy)-1-benzyl-2-ethyl-1H-indol-3-yl)-2-oxoacetamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Meng H, Liu Y, Zhai Y, Lai L. Optimization of 5-hydroxytryptamines as dual function inhibitors targeting phospholipase A2 and leukotriene A4 hydrolase. Eur J Med Chem. 2013 Jan;59:160-7
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