CPI-360( CPI-360 | CPI360 | CPI 360 )

Catalog No. M17382 CAS No. 1802175-06-9

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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Product Name

CPI-360
Note

Research use only, not for human use.
Brief Description

CPI-360 is a potent, selective, and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM, >100-fold selectivity over other methyltransferases.
Description

CPI-360 is a potent, selective,and SAM-competitive EZH1 inhibitor with IC50 of 102.3 nM
In Vitro

——
In Vivo

——
Synonyms

CPI-360 | CPI360 | CPI 360
Pathway

Others
Target

Other Targets
Recptor

EZH1
Research Area

Cancer
Indication

——

CAS Number

1802175-06-9
Formula Weight

437.53
Molecular Formula

C25H31N3O4
Purity

>98% (HPLC)
Solubility

DMSO : ≥ 48.9 mg/mL; 111.76 mM
SMILES

COC1=C(CNC(=O)C2=C(C)N([C@H](C)C3CCOCC3)C3=C2C=CC=C3)C(=O)NC(C)=C1
Chemical Name

(R)-N-((4-methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(tetrahydro-2H-pyran-4-yl)ethyl)-1H-indole-3-carboxamide