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CZC-8004
CAS No. 916603-07-1
CZC-8004( CZC 8004 | CZC8004 | Dianilinopyrimidine-01 )
Catalog No. M16584 CAS No. 916603-07-1
CZC-8004 (CZC8004, Dianilinopyrimidine-01) is a pan-specific kinase inhibitor that binds to a broad range of tyrosine kinases.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 80 | In Stock |
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| 10MG | 132 | In Stock |
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| 25MG | 282 | In Stock |
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| 50MG | 421 | In Stock |
|
| 100MG | 606 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCZC-8004
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NoteResearch use only, not for human use.
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Brief DescriptionCZC-8004 (CZC8004, Dianilinopyrimidine-01) is a pan-specific kinase inhibitor that binds to a broad range of tyrosine kinases.
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DescriptionCZC-8004 (CZC8004, Dianilinopyrimidine-01) is a pan-specific kinase inhibitor that binds to a broad range of tyrosine kinases, including ABL, BTK, FAK, FER, JAK1, SRC, SYK, TEC, TNK1, TYK2, and YES at low micromolar concentrations.
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In Vitro——
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In Vivo——
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SynonymsCZC 8004 | CZC8004 | Dianilinopyrimidine-01
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PathwayAngiogenesis
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TargetBcr-Abl
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RecptorBcr-Abl
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Research Area——
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Indication——
Chemical Information
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CAS Number916603-07-1
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Formula Weight309.3
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Molecular FormulaC17H16FN5
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Purity>98% (HPLC)
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SolubilityDMSO : 77.5 mg/mL 250.53 mM
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SMILESC1=CC=C(C=C1)NC2=NC(=NC=C2F)NC3=CC=C(C=C3)CN
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Chemical NameN2-?[4-?(aminomethyl)?phenyl]?-?5-?fluoro-?N4-?phenyl-2,?4-?pyrimidinediamine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Klutchko SR, et al. J Med Chem. 1998 Aug 13;41(17):3276-92.
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