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Setiptiline maleate
CAS No. 85650-57-3
Setiptiline maleate( MO-8282 )
Catalog No. M16210 CAS No. 85650-57-3
A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 47 | In Stock |
|
| 10MG | 47 | In Stock |
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| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSetiptiline maleate
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NoteResearch use only, not for human use.
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Brief DescriptionA tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist.
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DescriptionA tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, as well as an H1 receptor inverse agonist/antihistamine.Depression Approved.
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In Vitro——
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In Vivo——
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SynonymsMO-8282
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PathwayGPCR/G Protein
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Target5-HT Receptor
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Recptor5-HT Receptor
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Research AreaNeurological Disease
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IndicationDepression
Chemical Information
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CAS Number85650-57-3
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Formula Weight377.433
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Molecular FormulaC23H23NO4
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESCN1CCC2=C(C1)C3=CC=CC=C3CC4=CC=CC=C24.C(=CC(=O)O)C(=O)O
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Chemical Name1H-Dibenzo[3,4:6,7]cyclohepta[1,2-c]pyridine, 2,3,4,9-tetrahydro-2-methyl-, (2Z)-2-butenedioate (1:1)
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Niho T, et al. Nihon Yakurigaku Zasshi. 1986 Oct;88(4):309-20.
2. Mizota M, et al. Nihon Yakurigaku Zasshi. 1986 Dec;88(6):457-66.
3. Przegaliński E, et al. Pol J Pharmacol Pharm. 1986 Jul-Aug;38(4):377-84.
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