SR-57227

CAS No. 77145-51-8

SR-57227( SR 57227 | SR57227 )

Catalog No. M15916 CAS No. 77145-51-8

SR-57227 is a high affinity, selective 5-HT3 receptor agonist, demonstrates anticonvulsant effects in vivo.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    SR-57227
  • Note
    Research use only, not for human use.
  • Brief Description
    SR-57227 is a high affinity, selective 5-HT3 receptor agonist, demonstrates anticonvulsant effects in vivo.
  • Description
    SR-57227 is a high affinity, selective 5-HT3 receptor agonist, demonstrates anticonvulsant effects in vivo.Depression Discontinued.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    SR 57227 | SR57227
  • Pathway
    GPCR/G Protein
  • Target
    5-HT Receptor
  • Recptor
    5-HT Receptor
  • Research Area
    Neurological Disease
  • Indication
    Depression

Chemical Information

  • CAS Number
    77145-51-8
  • Formula Weight
    211.693
  • Molecular Formula
    C10H14ClN3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    NC1CCN(C2=NC(Cl)=CC=C2)CC1
  • Chemical Name
    1-(6-Chloro-2-pyridinyl)-4-piperidinamine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Li B, et al. PLoS One. 2014 Apr 1;9(4):e93158. 2. Gholipour T, et al. Seizure. 2010 Jan;19(1):17-22. 3. Ortega JE, et al. Neuropharmacology. 2012 Jun;62(8):2472-9. 4. Guo W, et al. Mol Pain. 2014 Jun 9;10:35.
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