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CK1-IN-3c
CAS No. 756805-89-7
CK1-IN-3c( —— )
Catalog No. M15877 CAS No. 756805-89-7
CK1-IN-3c is a novel casein kinase 1δ/ε (CK1δ/ε) inhibitor with IC50 of 1.6 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameCK1-IN-3c
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NoteResearch use only, not for human use.
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Brief DescriptionCK1-IN-3c is a novel casein kinase 1δ/ε (CK1δ/ε) inhibitor with IC50 of 1.6 uM.
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DescriptionCK1-IN-3c is a novel casein kinase 1δ/ε (CK1δ/ε) inhibitor with IC50 of 1.6 uM; shows selectivity over CDK5/p25, GSK-3α/β, and DYRK1A; elicits selective cytotoxic activity against the PANC-1 cell line.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetCasein Kinase
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RecptorCasein Kinase
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Research Area——
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Indication——
Chemical Information
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CAS Number756805-89-7
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Formula Weight347.378
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Molecular FormulaC19H17N5O2
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name6,7-dimethoxy-N-(5-phenyl-1H-pyrazol-3-yl)quinazolin-4-amine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Karthikeyan C, et al. Bioorg Med Chem Lett. 2017 Jun 15;27(12):2663-2667.
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