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PPT
CAS No. 263717-53-9
PPT( PPT )
Catalog No. M13809 CAS No. 263717-53-9
An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 92 | In Stock |
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| 5MG | 85 | In Stock |
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| 10MG | 136 | In Stock |
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| 25MG | 264 | In Stock |
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| 50MG | 390 | In Stock |
|
| 100MG | 589 | In Stock |
|
| 200MG | 827 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePPT
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NoteResearch use only, not for human use.
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Brief DescriptionAn allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.
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DescriptionAn allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.
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In VitroThe EC50 of Propyl pyrazole triol for the ERα-dependent response is 140 pM in ERα-U2OS-Luc cells.
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In Vivo——
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SynonymsPPT
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PathwayMembrane Transporter/Ion Channel
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TargetGAT
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RecptorGAT
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Research Area——
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Indication——
Chemical Information
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CAS Number263717-53-9
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Formula Weight388.467
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Molecular FormulaC24H24N2O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : ≥ 100 mg/mL (258.77 mM)
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SMILESOC1=CC=C(C2=C(CCC)C(C3=CC=C(O)C=C3)=NN2C4=CC=C(O)C=C4)C=C1
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Chemical Name4,4',4″-(4-propyl-[1H]-pyrazole-1,3,5-triyl)trisphenol
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Yamaura K, et al. Nat Chem Biol. 2016 Oct;12(10):822-30.
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