CARM1 inhibitor 9

CAS No. 2180931-09-1

CARM1 inhibitor 9( —— )

Catalog No. M13481 CAS No. 2180931-09-1

CARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    CARM1 inhibitor 9
  • Note
    Research use only, not for human use.
  • Brief Description
    CARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM.
  • Description
    CARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM; displays 20-fold selective for CARM1 over PRMT6 and highly selective over PRMT1, PRMT3, PRMT8 as well as PRMT5 and PRMT7; CARM1 inhibitor 9 is a useful tool for studying the role of CARM1 in health and disease.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Chromatin/Epigenetic
  • Target
    HMTase
  • Recptor
    HMTase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2180931-09-1
  • Formula Weight
    326.282
  • Molecular Formula
    C15H24BrN3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    ——
  • Chemical Name
    N-(3-bromobenzyl)-1-(2-(methylamino)ethyl)piperidin-4-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Kaniskan Hü, et al. Medchemcomm. 2016 Sep 1;7(9):1793-1796.
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