SC-806
CAS No. 216505-89-4
SC-806( SC 806 | SC806 )
Catalog No. M13454 CAS No. 216505-89-4
A potent, orally active p38 MAPK inhibitor with IC50 of 50 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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| 100MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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Biological Information
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Product NameSC-806
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, orally active p38 MAPK inhibitor with IC50 of 50 nM.
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DescriptionA potent, orally active p38 MAPK inhibitor with IC50 of 50 nM, significantly decreases incidence of arthritis in mouse collagen-induced arthritis.
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In Vitro——
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In Vivo——
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SynonymsSC 806 | SC806
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PathwayMAPK/ERK Signaling
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Targetp38 MAPK
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Recptorp38 MAPK
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Research Area——
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Indication——
Chemical Information
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CAS Number216505-89-4
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Formula Weight353.854
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Molecular FormulaC19H20ClN5
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name1-(5-(4-chlorophenyl)-4-(4-pyridinyl)-1H-pyrazol-3-yl)-4-methylpiperazine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Graneto MJ, et al. J Med Chem. 2007 Nov 15;50(23):5712-9.
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