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Home - Products - Chromatin/Epigenetic - Histone Demethylase - LSD1-IN-11p

LSD1-IN-11p

CAS No. 2101951-67-9

LSD1-IN-11p( —— )

Catalog No. M13339 CAS No. 2101951-67-9

LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    LSD1-IN-11p
  • Note
    Research use only, not for human use.
  • Brief Description
    LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM.
  • Description
    LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Chromatin/Epigenetic
  • Target
    Histone Demethylase
  • Recptor
    Histone Demethylase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2101951-67-9
  • Formula Weight
    420.473
  • Molecular Formula
    C22H24N6O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    ——
  • Chemical Name
    (R)-4-(3-(3-aminopiperidine-1-carbonyl)-5-((3-ethylisoxazol-5-yl)methoxy)-1H-pyrazol-1-yl)benzonitrile

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Mould DP, et al. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3190-3195.
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