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PI3Kδ-IN-7n
CAS No. 2088525-31-7
PI3Kδ-IN-7n( —— )
Catalog No. M13260 CAS No. 2088525-31-7
PI3Kδ-IN-7n is a highly potent and selective PI3Kδ inhibitor with IC50 of 0.9 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 146 | In Stock |
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| 5MG | 289 | In Stock |
|
| 10MG | 226 | In Stock |
|
| 25MG | 372 | In Stock |
|
| 50MG | 498 | In Stock |
|
| 100MG | 681 | In Stock |
|
| 200MG | 917 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
| 5MG | 150 | In Stock |
|
| 10MG | 226 | In Stock |
|
| 25MG | 372 | In Stock |
|
| 50MG | 498 | In Stock |
|
| 100MG | 681 | In Stock |
|
| 200MG | 917 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePI3Kδ-IN-7n
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NoteResearch use only, not for human use.
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Brief DescriptionPI3Kδ-IN-7n is a highly potent and selective PI3Kδ inhibitor with IC50 of 0.9 nM.
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DescriptionPI3Kδ-IN-7n is a highly potent and selective PI3Kδ inhibitor with IC50 of 0.9 nM, displays high selectivity (>1,500-fold) over PI3Kα, PI3Kβ, PI3Kγ (IC50>1.5 uM); shows reasonable pharmacokinetics with good bioavailability and moderate in vivo half-life; one of the most selective PI3Kδ inhibitors published to date.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorPI3K
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Research Area——
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Indication——
Chemical Information
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CAS Number2088525-31-7
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Formula Weight429.459
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Molecular FormulaC23H20FN7O
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name4-(3-amino-6-(1-methyl-5-(1-phenylcyclopropyl)-1H-1,2,4-triazol-3-yl)pyrazin-2-yl)-2-fluorobenzamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Terstiege I, et al. Bioorg Med Chem Lett. 2017 Feb 1;27(3):679-687.
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