CN-SAH
CAS No. 1985669-27-9
CN-SAH( —— )
Catalog No. M13103 CAS No. 1985669-27-9
CN-SAH is a potent and selective inhibitor of histone methyl transferase DOT1L with IC50 of 26 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
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| 50MG | 1782 | Get Quote |
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| 100MG | 2250 | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameCN-SAH
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NoteResearch use only, not for human use.
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Brief DescriptionCN-SAH is a potent and selective inhibitor of histone methyl transferase DOT1L with IC50 of 26 nM.
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DescriptionCN-SAH is a potent and selective inhibitor of histone methyl transferase DOT1L with IC50 of 26 nM, displays >10-fold selectivity over DNMT1, PRMT3, PRMT5, and G9α.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorHMTase
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Research Area——
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Indication——
Chemical Information
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CAS Number1985669-27-9
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Formula Weight408.433
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Molecular FormulaC16H20N6O5S
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameS-(((2S,3R,4S,5R)-5-(4-amino-5-cyano-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl)-L-homocysteine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Spurr SS, et al. Bioorg Med Chem Lett. 2016 Sep 15;26(18):4518-22.
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