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Tadalafil
CAS No. 171596-29-5
Tadalafil( IC351, IC-351, IC 351, Tadalafil, Adcirca, Cialis )
Catalog No. M12614 CAS No. 171596-29-5
Tadalafil is a potent phosphodiesterase-5 (PDE5) inhibitor (IC50=1 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 48 | In Stock |
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| 10MG | 30 | In Stock |
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| 25MG | 48 | In Stock |
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| 50MG | 68 | In Stock |
|
| 100MG | 104 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 269 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTadalafil
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NoteResearch use only, not for human use.
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Brief DescriptionTadalafil is a potent phosphodiesterase-5 (PDE5) inhibitor (IC50=1 nM).
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DescriptionTadalafil is a potent phosphodiesterase-5 (PDE5) inhibitor (IC50=1 nM); no inhibition on most of the other families of PDEs, with the exception of PDE11.Sexual Dysfunction Approved.
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In Vitro——
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In Vivo——
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SynonymsIC351, IC-351, IC 351, Tadalafil, Adcirca, Cialis
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PathwayAngiogenesis
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TargetPDE
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RecptorPDE5
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Research AreaEndocrinology
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IndicationSexual Dysfunction
Chemical Information
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CAS Number171596-29-5
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Formula Weight389.404
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Molecular FormulaC22H19N3O4
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 52 mg/mL
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SMILESO=C([C@@]1([H])CC2=C([C@@H](C3=CC(OCO4)=C4C=C3)N15)NC6=C2C=CC=C6)N(C)CC5=O
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Chemical NamePyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione, 6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydro-2-methyl-, (6R,12aR)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Blount MA, et al. Mol Pharmacol, 2004, 66(1), 144-152.
2. Ring BJ, et al. Clin Pharmacol Ther, 2005, 77(1), 63-75.
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