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K-Ras G12C-IN-2
CAS No. 1629267-75-9
K-Ras G12C-IN-2( —— )
Catalog No. M12442 CAS No. 1629267-75-9
A novel and irreversible inhibitor of mutant K-ras G12C.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 662 | Get Quote |
|
| 50MG | 2142 | Get Quote |
|
| 100MG | 2790 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameK-Ras G12C-IN-2
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NoteResearch use only, not for human use.
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Brief DescriptionA novel and irreversible inhibitor of mutant K-ras G12C.
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DescriptionA novel and irreversible inhibitor of mutant K-ras G12C.
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In VitroK-Ras G12C-IN-2 is a covalent kras g12c inhibitor extracted from patent WO2014152588A1, compound V-35.
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In Vivo——
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Synonyms——
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PathwayMAPK/ERK Signaling
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TargetRas
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RecptorRas
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1629267-75-9
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Formula Weight418.9171
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Molecular FormulaC21H27ClN4O3
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 22 mg/mL
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SMILESC=CC(=O)N1CC(C1)N2CCN(CC2)C(=O)CNC3=C(C=C(C(=C3)C4CC4)Cl)O
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Chemical Name2-Propen-1-one, 1-[3-[4-[2-[(4-chloro-5-cyclopropyl-2-hydroxyphenyl)amino]acetyl]-1-piperazinyl]-1-azetidinyl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. From PCT Int. Appl. (2014), WO 2014152588 A1 20140925.
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