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K-Ras G12C-IN-1
CAS No. 1629265-17-3
K-Ras G12C-IN-1( —— )
Catalog No. M12441 CAS No. 1629265-17-3
A novel and irreversible inhibitor of mutant K-ras G12C.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 314 | Get Quote |
|
| 50MG | 1791 | Get Quote |
|
| 100MG | 3222 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameK-Ras G12C-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionA novel and irreversible inhibitor of mutant K-ras G12C.
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DescriptionA novel and irreversible inhibitor of mutant K-ras G12C.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMAPK/ERK Signaling
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TargetRas
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RecptorRas
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1629265-17-3
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Formula Weight448.3423
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Molecular FormulaC22H23Cl2N3O3
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 40 mg/mL
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SMILESCOC1=C(C=C(C(=C1)Cl)C2=CC=CC=C2Cl)NCC(=O)N3CCN(CC3)C(=O)C=C
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Chemical Name2-Propen-1-one, 1-[4-[2-[(2',6-dichloro-4-methoxy[1,1'-biphenyl]-3-yl)amino]acetyl]-1-piperazinyl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. From PCT Int. Appl. (2014), WO 2014152588 A1 20140925.
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