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LLY-2707
CAS No. 1621865-33-5
LLY-2707( LLY 2707 | LLY2707 )
Catalog No. M12388 CAS No. 1621865-33-5
LLY-2707 (LLY 2707, LLY2707) is a novel potent, selective, nonsteroidal glucocorticoid receptor antagonist with Ki of 2.13 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameLLY-2707
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NoteResearch use only, not for human use.
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Brief DescriptionLLY-2707 (LLY 2707, LLY2707) is a novel potent, selective, nonsteroidal glucocorticoid receptor antagonist with Ki of 2.13 nM.
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DescriptionLLY-2707 (LLY 2707, LLY2707) is a novel potent, selective, nonsteroidal glucocorticoid receptor antagonist with Ki of 2.13 nM; shows substantially lower potency at the other steroid receptors (AR, MR and PR); suppress amphetamine-induced increases in locomotor activity, reduces atypical antipsychotic-associated weight gain in rats.
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In Vitro——
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In Vivo——
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SynonymsLLY 2707 | LLY2707
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PathwayEndocrinology/Hormones
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TargetGR
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RecptorGR
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Research Area——
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Indication——
Chemical Information
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CAS Number1621865-33-5
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Formula Weight389.489
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Molecular FormulaC20H24FN3O2S
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameN-(5-(tert-butyl)-3-(2-fluoro-5-methylpyridin-4-yl)-2-methyl-1H-indol-7-yl)methanesulfonamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Sindelar DK, et al. J Pharmacol Exp Ther. 2014 Jan;348(1):192-201.
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