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Omuralide
CAS No. 154226-60-5
Omuralide( Clasto-lactacystin )
Catalog No. M12183 CAS No. 154226-60-5
A potent 20S proteasome inhibitor with IC50 of 49 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameOmuralide
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NoteResearch use only, not for human use.
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Brief DescriptionA potent 20S proteasome inhibitor with IC50 of 49 nM.
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DescriptionA potent 20S proteasome inhibitor with IC50 of 49 nM (inhibition of proteasomal chymotrypsin-like proteolytic activity).
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In Vitro——
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In Vivo——
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SynonymsClasto-lactacystin
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PathwayProteasome/Ubiquitin
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TargetProteasome
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RecptorProteasome
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number154226-60-5
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Formula Weight213.233
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Molecular FormulaC10H15NO4
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(N[C@@]12[C@@H](O)C(C)C)[C@H](C)[C@]2([H])OC1=O
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Chemical Name(1R,4R,5S)-1-[(1S)-1-Hydroxy-2-methylpropyl]-4-methyl-6-oxa-2-azabicyclo[3.2.0]heptane-3,7-dione
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Corey EJ, et al. Chem Pharm Bull (Tokyo). 1999 Jan;47(1):1-10.
2. List A, et al. Angew Chem Int Ed Engl. 2014 Jan 7;53(2):571-4.
3. Feling RH, et al. Angew Chem Int Ed Engl. 2003 Jan 20;42(3):355-7.
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