TAK-875 hemihydrate

CAS No. 1374598-80-7

TAK-875 hemihydrate( —— )

Catalog No. M11546 CAS No. 1374598-80-7

Fasiglifam (TAK-875) is a selective GPR40 agonist with EC50 of 14 nM in human GPR40 expressing CHO cell line.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 209 Get Quote
10MG 290 Get Quote
25MG 521 Get Quote
50MG 782 Get Quote
100MG Get Quote Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    TAK-875 hemihydrate
  • Note
    Research use only, not for human use.
  • Brief Description
    Fasiglifam (TAK-875) is a selective GPR40 agonist with EC50 of 14 nM in human GPR40 expressing CHO cell line.
  • Description
    Fasiglifam (TAK-875) is a selective GPR40 agonist with EC50 of 14 nM in human GPR40 expressing CHO cell line, 400-fold more potent than oleic acid.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    GPR
  • Recptor
    GPR40
  • Research Area
    Metabolic Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    1374598-80-7
  • Formula Weight
    533.63
  • Molecular Formula
    C29H32O7S.1/2H2O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:93 mg/mL (174.3 mM);Ethanol:<1 mg/mL;Water:<1 mg/mL
  • SMILES
    O=C(O)C[C@@H]1COC2=CC(OCC3=CC(C4=C(C)C=C(OCCCS(=O)(C)=O)C=C4C)=CC=C3)=CC=C12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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