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TAK1-IN-1
CAS No. 1356013-39-2
TAK1-IN-1( —— )
Catalog No. M11459 CAS No. 1356013-39-2
TAK1-IN-1 is a potent, selective, Type I (ATP-competitive, DFG-in) TAK1 inhibitor with Kd of 59 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameTAK1-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionTAK1-IN-1 is a potent, selective, Type I (ATP-competitive, DFG-in) TAK1 inhibitor with Kd of 59 nM.
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DescriptionTAK1-IN-1 is a potent, selective, Type I (ATP-competitive, DFG-in) TAK1 inhibitor with Kd of 59 nM, a thienopyrimidine scaffold that serves as a good starting point for medicinal chemistry.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayNF-κB
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TargetTAK1
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RecptorTAK1
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Research Area——
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Indication——
Chemical Information
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CAS Number1356013-39-2
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Formula Weight336.369
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Molecular FormulaC17H12N4O2S
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameN-(7-methoxyquinolin-6-yl)thieno[3,2-d]pyrimidine-7-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Miura T, et al. Bioorg Med Chem Lett. 2017 Feb 15;27(4):1031-1036.
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