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IDH1-IN-1
CAS No. 1355326-21-4
IDH1-IN-1( Mutant IDH1-IN-1 )
Catalog No. M11452 CAS No. 1355326-21-4
Mutant IDH1-IN-1 is a potent mutant IDH1 R132H inhibitor with IC50 < 0.1 uM(A level in Patent).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 65 | In Stock |
|
| 2MG | 37 | In Stock |
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| 5MG | 62 | In Stock |
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| 10MG | 95 | In Stock |
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| 25MG | 183 | In Stock |
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| 50MG | 257 | In Stock |
|
| 100MG | 375 | In Stock |
|
| 200MG | 507 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameIDH1-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionMutant IDH1-IN-1 is a potent mutant IDH1 R132H inhibitor with IC50 < 0.1 uM(A level in Patent).
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DescriptionMutant IDH1-IN-1 is a potent mutant IDH1 R132H inhibitor with IC50 < 0.1 uM(A level in Patent); more bioactivity information in Patent WO2012009678A1(Example 135).
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In Vitro——
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In Vivo——
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SynonymsMutant IDH1-IN-1
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PathwayMetabolic Enzyme/Protease
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TargetDehydrogenase
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Recptormutant IDH1 R132H
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1355326-21-4
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Formula Weight498.59
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Molecular FormulaC30H31FN4O2
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Purity>98% (HPLC)
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SolubilityDMSO: 10 mM
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SMILESO=C(NC1CCCCC1)C(N(C(CN2C3=CC=CC=C3N=C2)=O)C4=CC=CC(F)=C4)C5=CC=CC=C5C
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Chemical Name2-(N-[2-(Benzimidazol-1-yl)acetyl]-3-fluoroanilino)-N-cyclohexyl-2-(2-methylphenyl)acetamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Janeta Popovici-Muller, et al. Patent WO2012009678 A
molnova catalog
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Mutant IDH1 inhibito...
Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).
