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BI 187004
CAS No. 1303515-32-3
BI 187004( BI187004 | VTP-34072 )
Catalog No. M11216 CAS No. 1303515-32-3
BI 187004 (VTP-34072) is a novel potent, selective 11β-hydroxysteroid dehydrogenase 1 (11β-HSD1) inhibitor intended to treat type 2 diabetes mellitus (T2D).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 206 | Get Quote |
|
| 10MG | 371 | Get Quote |
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| 25MG | 617 | Get Quote |
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| 50MG | 879 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameBI 187004
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NoteResearch use only, not for human use.
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Brief DescriptionBI 187004 (VTP-34072) is a novel potent, selective 11β-hydroxysteroid dehydrogenase 1 (11β-HSD1) inhibitor intended to treat type 2 diabetes mellitus (T2D).
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DescriptionBI 187004 (VTP-34072) is a novel potent, selective 11β-hydroxysteroid dehydrogenase 1 (11β-HSD1) inhibitor intended to treat type 2 diabetes mellitus (T2D).Diabetes Phase 2 Discontinued.
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In Vitro——
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In Vivo——
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SynonymsBI187004 | VTP-34072
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PathwayMetabolic Enzyme/Protease
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Target11β-HSD
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Recptor11β-HSD
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Research AreaMetabolic Disease
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IndicationDiabetes
Chemical Information
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CAS Number1303515-32-3
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Formula Weight342.402
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Molecular FormulaC21H18N4O
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name(4aR,9aS)-1-(1H-benzo[d]imidazole-5-carbonyl)-2,3,4,4a,9,9a-hexahydro1H-indeno[2,1-b]pyridine-6-carbonitrile
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Maw HH, et al. Drug Metab Dispos. 2018 Mar 7. pii: dmd.117.079764.
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