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BI 639667
CAS No. 1295298-26-8
BI 639667( BI639667 | BI-639667 )
Catalog No. M11194 CAS No. 1295298-26-8
BI 639667 (BI639667) is a potent and selective antagonist of human CCR1 with binding IC50 of 5.4 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 316 | In Stock |
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| 5MG | 281 | In Stock |
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| 10MG | 493 | In Stock |
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| 25MG | 924 | In Stock |
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| 50MG | 1311 | In Stock |
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| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBI 639667
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NoteResearch use only, not for human use.
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Brief DescriptionBI 639667 (BI639667) is a potent and selective antagonist of human CCR1 with binding IC50 of 5.4 nM.
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DescriptionBI 639667 (BI639667) is a potent and selective antagonist of human CCR1 with binding IC50 of 5.4 nM, inhibits chemotaxis with IC50 of 2.4 nM; shows good physico-chemical and pharmacokinetic properties.
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In Vitro——
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In Vivo——
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SynonymsBI639667 | BI-639667
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PathwayGPCR/G Protein
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TargetChemokine Receptor
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RecptorChemokine Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number1295298-26-8
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Formula Weight451.476
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Molecular FormulaC22H18FN5O3S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 10 mg/mL (22.15 mM)
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SMILESO=C(C1=CN=CC2=C1C=NN2C3=CC=C(F)C=C3)NC4(C5=CC(S(=O)(C)=O)=NC=C5)CC4
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Chemical Name1-(4-fluorophenyl)-N-(1-(2-(methylsulfonyl)pyridin-4-yl)cyclopropyl)-1H-pyrazolo[3,4-c]pyridine-4-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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