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N-desmethyl Enzalutamide
CAS No. 1242137-16-1
N-desmethyl Enzalutamide( N-desmethyl MDV3100 | N-desmethyl MDV 3100 | N-desmethyl MDV-3100 )
Catalog No. M10977 CAS No. 1242137-16-1
Amajor metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 50 | In Stock |
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| 2MG | 28 | In Stock |
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| 5MG | 46 | In Stock |
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| 10MG | 65 | In Stock |
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| 25MG | 133 | In Stock |
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| 50MG | 250 | In Stock |
|
| 100MG | 367 | In Stock |
|
| 200MG | 520 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameN-desmethyl Enzalutamide
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NoteResearch use only, not for human use.
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Brief DescriptionAmajor metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer.
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DescriptionAmajor metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer.
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In Vitro——
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In Vivo——
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SynonymsN-desmethyl MDV3100 | N-desmethyl MDV 3100 | N-desmethyl MDV-3100
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PathwayEndocrinology/Hormones
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TargetAndrogen Receptor (AR)
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RecptorAndrogen Receptor (AR)
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1242137-16-1
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Formula Weight450.4094
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Molecular FormulaC20H14F4N4O2S
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 48 mg/mL
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SMILESCC1(C(=O)N(C(=S)N1C2=CC(=C(C=C2)C(=O)N)F)C3=CC(=C(C=C3)C#N)C(F)(F)F)C
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Chemical NameBenzamide, 4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-thioxo-1-imidazolidinyl]-2-fluoro-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Tran C, et al. Science. 2009 May 8;324(5928):787-90.
2. Richards J, et al. Cancer Res. 2012 May 1;72(9):2176-82.
3. Gibbons JA, et al. Clin Pharmacokinet. 2015 Oct;54(10):1043-55.
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