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CaMKII-IN-1
CAS No. 1208123-85-6
CaMKII-IN-1( CaMKII-IN-1 | CaMKII | CaMKII IN-1 | CaMKII IN 1 )
Catalog No. M10773 CAS No. 1208123-85-6
A potent and highly selective CaMKII inhibitor with IC50 of 63 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 140 | In Stock |
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| 2MG | 65 | In Stock |
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| 5MG | 116 | In Stock |
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| 10MG | 169 | In Stock |
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| 25MG | 353 | In Stock |
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| 50MG | 538 | In Stock |
|
| 100MG | 775 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCaMKII-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionA potent and highly selective CaMKII inhibitor with IC50 of 63 nM.
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DescriptionA potent and highly selective CaMKII inhibitor with IC50 of 63 nM; no inhibitory effect for CaMKIV, MLCK, p38α, Akt1, PKC etc; shows 25-fold higher potency than KN-93.
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In Vitro——
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In Vivo——
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SynonymsCaMKII-IN-1 | CaMKII | CaMKII IN-1 | CaMKII IN 1
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PathwayEndocrinology/Hormones
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TargetCaMK
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RecptorCaMK
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number1208123-85-6
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Formula Weight548.0988
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Molecular FormulaC29H30ClN5O2S
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 54 mg/mL
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SMILESO=S(C1=CC=CC(Cl)=C1C)(NC2=C(CN(CC3=CC=CC=C3)CC4)C4=NC(NCCC5=CC=CC=C5)=N2)=O
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Chemical NameBenzenesulfonamide, 3-chloro-2-methyl-N-[5,6,7,8-tetrahydro-2-[(2-phenylethyl)amino]-6-(phenylmethyl)pyrido[4,3-d]pyrimidin-4-yl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Asano S, et al. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6696-8.
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