AM-0216

CAS No. 1202764-61-1

AM-0216( AM0216 )

Catalog No. M10737 CAS No. 1202764-61-1

AM-0216 (AM0216) is a highly potent inhibitor of NF-κB inducing Kinase (NIK).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    AM-0216
  • Note
    Research use only, not for human use.
  • Brief Description
    AM-0216 (AM0216) is a highly potent inhibitor of NF-κB inducing Kinase (NIK).
  • Description
    AM-0216 (AM0216) is a highly potent inhibitor of NF-κB inducing Kinase (NIK), example 294 in patent WO 2009158011 A1.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    AM0216
  • Pathway
    Apoptosis
  • Target
    NF-κB
  • Recptor
    NF-κB
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1202764-61-1
  • Formula Weight
    363.439
  • Molecular Formula
    C19H17N5OS
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(C#CC1=CC2=C(CCN2C3=NC(=NC=C3)N)C=C1)(C4=NC=CS4)O
  • Chemical Name
    (R)-4-(1-(2-aminopyrimidin-4-yl)indolin-6-yl)-2-(thiazol-2-yl)but-3-yn-2-ol

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Henry KL, et al. Sci Signal. 2018 Jul 31;11(541). pii: eaam8216. 2. Example 294 in patent WO 2009158011 A1.
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