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Rapastinel
CAS No. 117928-94-6
Rapastinel( GLYX-13 | Thr-Pro-Pro-Thr-NH2 )
Catalog No. M10606 CAS No. 117928-94-6
A tetrapeptide (TPPT-amide) that acts as a NMDA receptor glycine site partial agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 78 | In Stock |
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| 2MG | 46 | In Stock |
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| 5MG | 73 | In Stock |
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| 10MG | 111 | In Stock |
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| 25MG | 188 | In Stock |
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| 50MG | 334 | In Stock |
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| 100MG | 496 | In Stock |
|
| 200MG | 715 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRapastinel
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NoteResearch use only, not for human use.
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Brief DescriptionA tetrapeptide (TPPT-amide) that acts as a NMDA receptor glycine site partial agonist.
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DescriptionA tetrapeptide (TPPT-amide) that acts as a NMDA receptor glycine site partial agonist; readily crosses the blood-brain barrier and modulates the NMDA receptor, shows potent cognitive-enhancing properties in a valid in vivo model of learning.Depression Phase 3 Clinical.
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In Vitro——
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In Vivo——
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SynonymsGLYX-13 | Thr-Pro-Pro-Thr-NH2
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PathwayMembrane Transporter/Ion Channel
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TargetiGluR
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RecptorOthers
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Research AreaNeurological Disease
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IndicationDepression
Chemical Information
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CAS Number117928-94-6
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Formula Weight413.4686
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Molecular FormulaC18H31N5O6
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 32 mg/mL
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SMILESC[C@@H](O)[C@@H](C(N)=O)NC([C@H]1N(C([C@H]2N(C([C@H]([C@H](O)C)N)=O)CCC2)=O)CCC1)=O
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Chemical NameL-Threoninamide, L-threonyl-L-prolyl-L-prolyl-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Moskal JR, et al. Neuropharmacology. 2005 Dec;49(7):1077-87.
2. Zhang XL, et al. Neuropharmacology. 2008 Dec;55(7):1238-50.
3. Burgdorf J, et al. Neurobiol Aging. 2011 Apr;32(4):698-706.
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