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CI-976
CAS No. 114289-47-3
CI-976( PD 128042 )
Catalog No. M10507 CAS No. 114289-47-3
CI-976 (PD 128042) is a potent, selective, orally bioavailable inhibitor of ACAT-1 (Acetyl-CoA acetyltransferase 1) with IC50 of 73 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 88 | In Stock |
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| 5MG | 56 | In Stock |
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| 10MG | 105 | In Stock |
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| 25MG | 231 | In Stock |
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| 50MG | 379 | In Stock |
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| 100MG | 630 | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCI-976
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NoteResearch use only, not for human use.
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Brief DescriptionCI-976 (PD 128042) is a potent, selective, orally bioavailable inhibitor of ACAT-1 (Acetyl-CoA acetyltransferase 1) with IC50 of 73 nM.
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DescriptionCI-976 (PD 128042) is a potent, selective, orally bioavailable inhibitor of ACAT-1 (Acetyl-CoA acetyltransferase 1) with IC50 of 73 nM; decreases plasma total cholesterol, very low density lipoprotein (VLDL) cholesterol, LDL cholesterol, apolipoprotein B, liver cholesteryl esters, and VLDL and LDL cholesteryl ester content in rabbits.Atherosclerosis Discontinued.
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In Vitro——
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In Vivo——
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SynonymsPD 128042
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PathwayOthers
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TargetOther Targets
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RecptorOther Targets
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Research AreaCardiovascular Disease
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IndicationAtherosclerosis
Chemical Information
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CAS Number114289-47-3
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Formula Weight393.568
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Molecular FormulaC23H39NO4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (254.09 mM)
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SMILESCCCCCCCCCCC(C)(C)C(=O)NC1=C(C=C(C=C1OC)OC)OC
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Chemical Name2,2-dimethyl-N-(2,4,6-trimethoxyphenyl)-dodecanamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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Aerugidiol
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γ-2-MSH (41-58), ami...
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