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PV-1115
CAS No. 1093793-10-2
PV-1115( PV 1115 | PV1115 )
Catalog No. M10360 CAS No. 1093793-10-2
A potent and highly selective Chk2 inhibitor with IC50 of 0.14 nM; displays greater than 100 uM for Chk1 in vitro.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NamePV-1115
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NoteResearch use only, not for human use.
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Brief DescriptionA potent and highly selective Chk2 inhibitor with IC50 of 0.14 nM; displays greater than 100 uM for Chk1 in vitro.
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DescriptionA potent and highly selective Chk2 inhibitor with IC50 of 0.14 nM; displays greater than 100 uM for Chk1 in vitro.
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In Vitro——
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In Vivo——
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SynonymsPV 1115 | PV1115
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PathwayAngiogenesis
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TargetChk
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RecptorChk
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Research Area——
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Indication——
Chemical Information
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CAS Number1093793-10-2
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Formula Weight405.418
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Molecular FormulaC20H19N7O3
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(C(N1)=CC2=C1C([N+]([O-])=O)=CC=C2)NC3=CC=C(/C(C)=N/NC4=NCCN4)C=C3
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Chemical NameN-(4-(1-(2-(4,5-dihydro-1H-imidazol-2-yl)hydrazono)ethyl)phenyl)-7-nitro-1H-indole-2-carboxamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Lountos GT, et al. J Struct Biol. 2011 Dec; 176(3):292-301.
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