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Pim1/AKK1-IN-1
CAS No. 1093222-27-5
Pim1/AKK1-IN-1( LKB1/AAK1 dual inhibitor )
Catalog No. M10359 CAS No. 1093222-27-5
A potent, multikinase inhibitor and also inhibits MPSK1 and TNIK.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 120 | In Stock |
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| 5MG | 174 | In Stock |
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| 10MG | 263 | In Stock |
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| 25MG | 464 | In Stock |
|
| 50MG | 672 | In Stock |
|
| 100MG | 945 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePim1/AKK1-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, multikinase inhibitor and also inhibits MPSK1 and TNIK.
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DescriptionA potent, multikinase inhibitor with Kd of 35/53/75/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and also inhibits MPSK1 and TNIK.
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In Vitro——
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In Vivo——
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SynonymsLKB1/AAK1 dual inhibitor
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PathwayJAK/STAT Signaling
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TargetPim
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RecptorPim
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1093222-27-5
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Formula Weight339.3501
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Molecular FormulaC20H13N5O
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=C(C1=CC=CN=C1)NC2=CNC3=NC=C(C4=CC=C(C#N)C=C4)C=C32
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Chemical Name3-Pyridinecarboxamide, N-[5-(4-cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Bamborough P, et al. J Med Chem. 2008 Dec 25;51(24):7898-914.
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