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GSK-3117391
CAS No. 1018673-42-1
GSK-3117391( CHR-5154 | GSK3117391 | CHR5154 )
Catalog No. M10089 CAS No. 1018673-42-1
GSK-3117391 (CHR-5154) is a novel macrophage-targeted HDAC inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 93 | In Stock |
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| 5MG | 85 | In Stock |
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| 10MG | 140 | In Stock |
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| 25MG | 282 | In Stock |
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| 50MG | 445 | In Stock |
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| 100MG | 714 | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGSK-3117391
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NoteResearch use only, not for human use.
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Brief DescriptionGSK-3117391 (CHR-5154) is a novel macrophage-targeted HDAC inhibitor.
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DescriptionGSK-3117391 (CHR-5154) is a novel macrophage-targeted HDAC inhibitor, has the potential to complement existing therapies in the treatment of chronic inflammatory disorders such as rheumatoid arthritis.Rheumatoid Arthritis Phase 2 Clinical.
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In Vitro——
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In Vivo——
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SynonymsCHR-5154 | GSK3117391 | CHR5154
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PathwayCell Cycle/DNA Damage
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TargetHDAC
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RecptorHDAC
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Research AreaInflammation/Immunology
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IndicationRheumatoid Arthritis
Chemical Information
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CAS Number1018673-42-1
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Formula Weight389.496
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Molecular FormulaC21H31N3O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (123.91 mM)
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SMILESO=C(OC1CCCC1)[C@H](C2CCCCC2)NCC3=CC=C(CCC(NO)=O)N=C3
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Chemical Namecyclopentyl (S)-2-cyclohexyl-2-((6-(3-(hydroxyamino)-3-oxopropyl)pyridin-3-yl)amino)acetate
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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