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Desloratadine
CAS No. 100643-71-8
Desloratadine( Descarboethoxyloratadine | NSC 675447 | SCH 34117 )
Catalog No. M10053 CAS No. 100643-71-8
Desloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 28 | In Stock |
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| 50MG | 32 | In Stock |
|
| 100MG | 55 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDesloratadine
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NoteResearch use only, not for human use.
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Brief DescriptionDesloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM.
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DescriptionDesloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM.
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In Vitro——
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In Vivo——
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SynonymsDescarboethoxyloratadine | NSC 675447 | SCH 34117
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorH1 receptor
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number100643-71-8
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Formula Weight310.82
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Molecular FormulaC19H19ClN2
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Purity>98% (HPLC)
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SolubilityEthanol: 62 mg/mL (199.47 mM); DMSO: 26 mg/mL (83.64 mM)
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SMILESC1CC2=C(C=CC(=C2)Cl)C(=C3CCNCC3)C4=C1C=CC=N4
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Chemical Name8-chloro-6,11-dihydro-11-(4-piperdinylidene)- 5h-benzo[5,6]cyclohepta[1,2-b]pyridine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Geha RS, et al. J Allergy Clin Immunol, 2001, 107(4), 751-762.
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