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Luzindole
CAS No. 117946-91-5
Luzindole ( N-0774 )
Catalog No. M23346 CAS No. 117946-91-5
Luzindole is a selective melatonin receptor antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 132 | In Stock |
|
| 10MG | 224 | In Stock |
|
| 25MG | 377 | In Stock |
|
| 50MG | 556 | In Stock |
|
| 100MG | 788 | In Stock |
|
| 500MG | 1575 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLuzindole
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NoteResearch use only, not for human use.
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Brief DescriptionLuzindole is a selective melatonin receptor antagonist.
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DescriptionLuzindole is a selective melatonin receptor antagonist. Luzindole inhibits experimental autoimmune encephalomyelitis and exerts antidepressant-like activity. Luzindole preferentially targets MT2 (Mel1b) over MT1 (Mel1a) with Ki values of 10.2 and 158 nM for human MT2 and MT1, respectively.
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SynonymsN-0774
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PathwayOthers
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TargetOther Targets
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RecptorMT1 receptor;MT2 receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number117946-91-5
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Formula Weight292.4
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Molecular FormulaC19H20N2O
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Purity>98% (HPLC)
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SolubilityDMSO:100 mg/mL (342.03 mM; Need ultrasonic)
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SMILESCC(NCCc1c(Cc2ccccc2)[nH]c2c1cccc2)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Dubocovich ML, et al. Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355(3):365-75.
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