LY2119620

CAS No. 886047-22-9

LY2119620 ( LY2119620; LY 2119620; LY-2119620 )

Catalog No. M17642 CAS No. 886047-22-9

LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 66 In Stock
5MG 113 In Stock
10MG 178 In Stock
25MG 344 In Stock
50MG 512 In Stock
100MG 737 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    LY2119620
  • Note
    Research use only, not for human use.
  • Brief Description
    LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.
  • Description
    LY2119620 is a positive allosteric modulator of the M2 and M4 muscarinic acetylcholine receptors (mAChRs).
  • Synonyms
    LY2119620; LY 2119620; LY-2119620
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    M2 mAChR;M4 mAChR
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    886047-22-9
  • Formula Weight
    437.94
  • Molecular Formula
    C19H24ClN5O3S
  • Purity
    98%
  • Solubility
    DMSO : 67.5 mg/mL. 154.13 mM; H2O : < 0.1 mg/mL
  • SMILES
    CN1CCN(CC1)C(=O)COc1nc2sc(C(=O)NC3CC3)c(N)c2c(C)c1Cl
  • Chemical Name
    3-amino-5-chloro-N-cyclopropyl-4-methyl-6-[2-(4-methyl-1-piperazinyl)-2-oxoethoxy]-thieno[2,3-b]pyridine-2-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Croy C H, Schober D A, Xiao H, et al. Characterization of the novel positive allosteric modulator, LY2119620, at the muscarinic M(2) and M(4) receptors.[J]. Molecular Pharmacology, 2014, 86(1):106-115.
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