LP-211

CAS No. 1052147-86-0

LP-211 ( —— )

Catalog No. M20108 CAS No. 1052147-86-0

LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 35 In Stock
5MG 58 In Stock
10MG 87 In Stock
25MG 170 In Stock
50MG 290 In Stock
100MG 462 In Stock
200MG 659 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    LP-211
  • Note
    Research use only not for human use.
  • Brief Description
    LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.
  • Description
    LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM) and >300-fold selectivity over the 5-HT1A receptor.
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT7;D2 receptor;5-HT1A receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1052147-86-0
  • Formula Weight
    466.62
  • Molecular Formula
    C30H34N4O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 90 mg/mL (192.87 mM)
  • SMILES
    O=C(CCCCCN1CCN(CC1)c1ccccc1-c1ccccc1)NCc1ccc(cc1)C#N
  • Chemical Name
    N-[(4-cyanophenyl)methyl]-6-[4-(2-phenylphenyl)piperazin-1-yl]hexanamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Leopoldo M et al. Structural modifications of N-(1234-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinehexanamides: influence on lipophilicity and 5-HT7 receptor activity. Part III. J Med Chem. 2008 Sep 25;51(18):5813-22.
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