LJ570
CAS No. 2252488-69-8
LJ570( —— )
Catalog No. M21635 CAS No. 2252488-69-8
LJ570 is the first PPARα/γ dual agonist (PPARαPPARγ with EC50s of 1.05 and 0.12 μM respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 338 | Get Quote |
|
| 5MG | 519 | Get Quote |
|
| 10MG | 743 | Get Quote |
|
| 25MG | 1134 | Get Quote |
|
| 50MG | 1512 | Get Quote |
|
| 100MG | 2061 | Get Quote |
|
| 500MG | 4131 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameLJ570
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NoteResearch use only, not for human use.
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Brief DescriptionLJ570 is the first PPARα/γ dual agonist (PPARαPPARγ with EC50s of 1.05 and 0.12 μM respectively.
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DescriptionLJ570 is the first PPARα/γ dual agonist (PPARαPPARγ with EC50s of 1.05 and 0.12 μM respectively)
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetPPAR
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RecptorPPAR
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Research Area——
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Indication——
Chemical Information
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CAS Number2252488-69-8
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Formula Weight394.5
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Molecular FormulaC27H22O3?
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Antonio L Luca P Carmen C et al. Identification of the First PPARα/γ Dual Agonist Able to Bind to Canonical and Alternate Sites of PPARγ and to Inhibit its Cdk5-Mediated Phosphorylation[J]. Journal of Medicinal Chemistry 2018:acs.jmedchem.8b00835-.
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