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LGD-4033
CAS No. 1165910-22-4
LGD-4033( LGD 4033 | LGD4033 | VK-5211 )
Catalog No. M10567 CAS No. 1165910-22-4
A novel nonsteroidal, oral selective androgen receptor modulator (SARM), binds androgen receptor with high affinity (Ki=1 nM) and selectivity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameLGD-4033
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NoteResearch use only, not for human use.
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Brief DescriptionA novel nonsteroidal, oral selective androgen receptor modulator (SARM), binds androgen receptor with high affinity (Ki=1 nM) and selectivity.
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DescriptionA novel nonsteroidal, oral selective androgen receptor modulator (SARM), binds androgen receptor with high affinity (Ki=1 nM) and selectivity; has favorable pharmacokinetic profile, and increases lean body mass even during this short period without change in prostate-specific antigen.Other Indication Phase 2 Clinical.
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In Vitro——
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In Vivo——
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SynonymsLGD 4033 | LGD4033 | VK-5211
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PathwayEndocrinology/Hormones
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TargetAndrogen Receptor (AR)
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RecptorAndrogen Receptor (AR)
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Research AreaOther Indications
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IndicationOther Disease
Chemical Information
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CAS Number1165910-22-4
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Formula Weight338.25
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Molecular FormulaC14H12F6N2O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : ≥ 100 mg/mL (295.64 mM)
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SMILESN#CC1=CC=C(N2[C@@H]([C@@H](O)C(F)(F)F)CCC2)C=C1C(F)(F)F
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Chemical Name4-((R)-2-((R)-2,2,2-trifluoro-1-hydroxyethyl)pyrrolidin-1-yl)-2-(trifluoromethyl)benzonitrile
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Basaria S, et al. J Gerontol A Biol Sci Med Sci. 2013 Jan;68(1):87-95.
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