LEE011

CAS No. 1211441-98-3

LEE011 ( Ribociclib )

Catalog No. M10790 CAS No. 1211441-98-3

LEE011 is an orally available, and highly specific CDK4/6 inhibitor. Phase 3.

Purity : >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 32 In Stock
5MG 53 In Stock
10MG 73 In Stock
25MG 93 In Stock
50MG 107 In Stock
100MG 161 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    LEE011
  • Note
    Research use only, not for human use.
  • Brief Description
    LEE011 is an orally available, and highly specific CDK4/6 inhibitor. Phase 3.
  • Description
    LEE011 is an orally available, and highly specific CDK4/6 inhibitor. Phase 3.
  • Synonyms
    Ribociclib
  • Pathway
    Angiogenesis
  • Target
    CDK
  • Recptor
    CDK4
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1211441-98-3
  • Formula Weight
    434.54
  • Molecular Formula
    C23H30N8O
  • Purity
    >98%(HPLC)
  • Solubility
    DMSO: 7 mg/mL (16.1 mM)
  • SMILES
    CN(C)C(=O)C1=CC2=CN=C(NC3=NC=C(C=C3)N3CCNCC3)N=C2N1C1CCCC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Rader J, et al. Clin Y Res. 2013, 19(22), 6173-6182.
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